D-3263 hydrochloride
CAS No. 1008763-54-9
D-3263 hydrochloride ( D3263 HCl salt; EC D-3263 HCl )
产品货号. M26136 CAS No. 1008763-54-9
D-3263 hydrochloride is enteric-coated, orally bioavailable (transient receptor potential melatonin member 8) TRPM8 agonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥915 | 有现货 |
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10MG | ¥1442 | 有现货 |
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25MG | ¥2697 | 有现货 |
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50MG | ¥4528 | 有现货 |
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100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称D-3263 hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述D-3263 hydrochloride is enteric-coated, orally bioavailable (transient receptor potential melatonin member 8) TRPM8 agonist.
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产品描述D-3263 hydrochloride is enteric-coated, orally bioavailable (transient receptor potential melatonin member 8) TRPM8 agonist.(In Vitro):D-3263 hydrochloride binds and activates TRPM8, which may lead to increased entry of calcium and sodium; destruction of calcium and sodium homeostasis; induction of cell death in tumor cells expressing TRPM8. D-3263 hydrochloride may reduce the level of dihydrotestosterone (DHT), which may contribute to its inhibitory effect on prostate cancer and BPH.
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同义词D3263 HCl salt; EC D-3263 HCl
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通路Others
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靶点Other Targets
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受体GnRHR
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研究领域——
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适应症——
化学信息
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CAS Number1008763-54-9
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分子量410.0
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分子式C21H32ClN3O3
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纯度>98% (HPLC)
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溶解度——
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SMILESCl.COc1ccc2n(C(=O)[C@@H]3C[C@H](C)CC[C@H]3C(C)C)c(=O)n(CCN)c2c1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Ezzati M, Carr BR (2015).?"Elagolix, a novel, orally bioavailable GnRH antagonist under investigation for the treatment of endometriosis-related pain".?Womens Health (Lond).?11?(1): 19–28.
产品手册
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